Epiamastatin · HCl

Names

[ Name ]:
Epiamastatin · HCl

[Synonym ]:
H-(2R,3R)-AHMH-VAL-VAL-ASP-OH HCL
(2R,3R)-[3-AMINO-2-HYDROXY-5-METHYLHEXANOYL]-VAL-VAL-ASP-OH HCL
MFCD00070396
[(2R,3R)-3-AMINO-2-HYDROXY-5-METHYLHEXANOYL]-VAL-VAL-ASP HYDROCHLORIDE
(2R,3R)-AHMHA-Val-Val-Asp-OH HCl
(2R,3R)-AHMHA-Val-Val-Asp-OH
EPIAMASTATIN
EPIAMASTATIN HCL
Epiamastatin · HCl

Chemical & Physical Properties

[ Boiling Point ]:
808ºC at 760mmHg

[ Molecular Formula ]:
C₂₁H₃₉ClN₄O₈

[ Molecular Weight ]:
511.00900

[ Flash Point ]:
442.5ºC

[ Exact Mass ]:
510.24600

[ PSA ]:
208.15000

[ LogP ]:
1.72140

[ Vapour Pressure ]:
3.23E-30mmHg at 25°C

MSDS

Click to get detail MSDS

Safety Information

[ Personal Protective Equipment ]:
Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter

[ RIDADR ]:
NONH for all modes of transport

[ WGK Germany ]:
3

Articles

Inhibition of aminopeptidases by amastatin and bestatin derivatives. Effect of inhibitor structure on slow-binding processes.

J. Med. Chem. 27 , 417, (1984)

Amastatin [(2S,3R)-3-amino-2-hydroxy-5-methylhexanoyl-L-valyl-L-valyl-L- aspartic acid] and bestatin [(2S,3R)-3-amino-2-hydroxy-4-phenylbutanoyl-L-leucine] are slow-binding, competitive inhibitors of ...