Ketocaine

Names

[ Name ]:
Ketocaine

[Synonym ]:
2-<2-Diaethylamino-aethoxycarbonyl>-phenthiazin
o-(Diisopropylaminoethoxy)-butyrophenon
EINECS 214-131-8
10H-phenothiazine-2-carboxylic acid 2-diethylamino-ethyl ester
2-(N-Diisopropylaminoethoxy)-1-butyro-phenon
2-<2-Diisopropylamino-aethoxy>-butyrophenon
2-diethylaminoethyl 10H-phenothiazine-2-carboxylate
Ketocaine

Biological Activity

[Description]:

Ketocaine is a butyrophenone derivative, which possesses local anesthetic activity.

[Related Catalog]:

Signaling Pathways >> Others >> Others

Research Areas >> Others

[In Vitro]

Ketocaine modifies the oxygen consumption by tissues with prevailing anaerobic metabolism and to inhibit the mitotic activity of human lymphocytes in culture stimulated by phytohemagglutinin[1].

[References]

[1]. Galatulas I, et al. New alkylating agents: butyrophenone derivatives. Anticancer Res. 1986 Jul-Aug;6(4):853-5.

[Related Small Molecules]

Chemical & Physical Properties

[ Density]:
0.966g/cm3

[ Boiling Point ]:
386.3ºC at 760mmHg

[ Molecular Formula ]:
C₁₈H₂₉NO₂

[ Molecular Weight ]:
291.42800

[ Flash Point ]:
187.5ºC

[ Exact Mass ]:
291.22000

[ PSA ]:
29.54000

[ LogP ]:
4.16700

[ Vapour Pressure ]:
3.57E-06mmHg at 25°C

[ Index of Refraction ]:
1.497

[ Storage condition ]:
2-8℃

Safety Information

[ HS Code ]:
2922509090

Customs

[ HS Code ]: 2922509090

[ Summary ]:
2922509090. other amino-alcohol-phenols, amino-acid-phenols and other amino-compounds with oxygen function. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:30.0%