GPR4 antagonist 1
Names
[ CAS No. ]:
1197879-16-5
[ Name ]:
GPR4 antagonist 1
[Synonym ]:
2-Ethyl-3-{4-[(E)-3-(4-isopropyl-piperazin-1-yl)-propenyl]-benzyl}-5,7-dimethyl-3H-imidazo[4,5-b]pyridine
GPR4 RECEPTOR MODULATOR 46
Biological Activity
[Description]:
GPR4 antagonist 1 is a GPR4 antagonist, with an IC50 of 189 nM.
[Related Catalog]:
[Target]
IC50: 189 nM (GPR4)[1].
[References]
[Related Small Molecules]
Captisol
|
Cyclosporin A
|
H2DCFDA
|
0MPTP hydrochloride
|
GW4869
|
Etomoxir
|
TD139
|
Mitoquinone mesylate
|
GSK2795039
|
JC-1
|
BAPTA-AM
|
AP 20187
|
Setanaxib (GKT137831)
|
D-Luciferin
|
Crotaline
Chemical & Physical Properties
[ Molecular Formula ]:
C27H37N5
[ Molecular Weight ]:
431.61600
[ Exact Mass ]:
431.30500
[ PSA ]:
37.19000
[ LogP ]:
4.57380