Cav 2.2 blocker 2

Names

[ CAS No. ]:
1204535-44-3

[ Name ]:
Cav 2.2 blocker 2

Biological Activity

[Description]:

Cav 2.2 blocker 2 is a Cav2.2 calcium channel blocker extracted from patent WO2017046581A1, compound 1. Cav 2.2 blocker 2 can reverses hyperalgesia associated with an injury or inflammation in conjunction with the opioid[1].

[Related Catalog]:

Signaling Pathways >> Membrane Transporter/Ion Channel >> Calcium Channel

Research Areas >> Neurological Disease

[Target]

N-Type Ca2+ Channel

[In Vitro]

Cav 2.2 blocker 2 (compound 1) (1-10 mg/kg; p.o.) in conjunction with Morphine (0.3 mg/kg) reverses the complete freunds adjuvant (CFA) induced hyperalgesia in rats[1].

[References]

[1]. Ali Z, et, al. Composition comprising cav2.2 calcium channel blocker and opioid. WO2017046581A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₉H₂₀F₃N₃O₃S

[ Molecular Weight ]:
427.44

Cav 2.2 blocker 2

Names

Biological Activity

Chemical & Physical Properties

Related Compounds