SB 205607 dihydrobromide
Names
[ CAS No. ]:
1217628-73-3
[ Name ]:
SB 205607 dihydrobromide
[Synonym ]:
Phenol, 3-[(4aS,12aR)-1,3,4,5,12,12a-hexahydro-2-methylpyrido[3,4-b]acridin-4a(2H)-yl]-, hydrobromide (1:2)
3-[(4aS,12aR)-2-Methyl-1,3,4,5,12,12a-hexahydropyrido[3,4-b]acridin-4a(2H)-yl]phenol dihydrobromide
Biological Activity
[Description]:
A potent and selective δ-opioid receptor agonist that has high affinity and selectivity for the δ1 subtype with Ki of 1.12 nM; dispalys >1,000-fold selectivity over μOR and κOR; Pain Discontinued
[References]
References 1. Knapp RJ, et al. Eur J Pharmacol. 1995 Oct 15;291(2):129-34. 2. Tseng LF, et al. J Pharmacol Exp Ther. 1997 Feb;280(2):600-5. 3. Fusa K, et al. Neuroscience. 2005;130(3):745-55. View Related Products by Target Opioid Receptor Pain
Chemical & Physical Properties
[ Molecular Formula ]:
C23H24N2O.2HBr
[ Molecular Weight ]:
506.273
[ Exact Mass ]:
504.041168