TAK1-IN-1
Names
[ CAS No. ]:
1356013-39-2
[ Name ]:
TAK1-IN-1
Biological Activity
[Description]:
TAK1-IN-1 is a potent, selective, Type I (ATP-competitive, DFG-in) TAK1 inhibitor with Kd of 59 nM, a thienopyrimidine scaffold that serves as a good starting point for medicinal chemistry.
[References]
References 1. Miura T, et al. Bioorg Med Chem Lett. 2017 Feb 15;27(4):1031-1036. View Related Products by Target TAK1
Chemical & Physical Properties
[ Molecular Formula ]:
C17H12N4O2S
[ Molecular Weight ]:
336.369