Plasma kallikrein-IN-4

Names

[ CAS No. ]:
1357954-34-7

[ Name ]:
Plasma kallikrein-IN-4

Biological Activity

[Description]:

Plasma kallikrein-IN-4 (Example 153) is a plasma kallikrein inhibitor with an IC50 of 0.016 μM against human plasma kallikrein[1].

[Related Catalog]:

Signaling Pathways >> Metabolic Enzyme/Protease >> Ser/Thr Protease

Research Areas >> Cardiovascular Disease

Research Areas >> Inflammation/Immunology

[Target]

IC50: 0.016 μM (human plasma kallikrein)[1]

[References]

[1]. Trixi Brandl, et al. N-((6-amino-pyridin-3-yl)methyl)-heteroaryl-carboxamides as inhibitors of plasma kallikrein. Patent WO2012017020A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₂H₂₃N₇O

[ Molecular Weight ]:
401.46

Related Compounds