PI3K-IN-31
Names
[ CAS No. ]:
1359956-12-9
[ Name ]:
PI3K-IN-31
Biological Activity
[Description]:
PI3K-IN-31 (Compound 6b) is a potent PI3K inhibitor with IC50s of 3.7 nM, 74 nM, 14.6 nM, and 9.9 nM for PI3Kα, PI3Kβ, PI3Kγ, and PI3Kδ, respectively. PI3K-IN-31 has anticancer effects[1].
[Related Catalog]:
[Target]
PI3Kα:3.7 nM (IC50)
PI3Kδ:9.9 nM (IC50)
PI3Kγ:14.6 nM (IC50)
PI3Kβ:74 nM (IC50)
[References]
Chemical & Physical Properties
[ Molecular Formula ]:
C19H23F2N7O3
[ Molecular Weight ]:
435.43