ZINC-3573 racemate
Names
[ CAS No. ]:
1378183-16-4
[ Name ]:
ZINC-3573 racemate
Biological Activity
[Description]:
ZINC-3573 racemate is a potent, selective agonist of the atypical opioid receptor MRGPRX2 (EC50=3 uM), showing little activity against 315 other GPCRs and 97 representative kinases; activates endogenous MRGPRX2 in a human mast cell line, inducing degranulation and calcium release.
[References]
References 1. Lansu K, et al. Nat Chem Biol. 2017 May;13(5):529-536. View Related Products by Target Other Targets
Chemical & Physical Properties
[ Molecular Formula ]:
C18H21N5
[ Molecular Weight ]:
307.401