BET bromodomain inhibitor
Names
[ CAS No. ]:
1505453-59-7
[ Name ]:
BET bromodomain inhibitor
[Synonym ]:
BETbromodomaininhibitor
BET bromodomain inhibitor
Biological Activity
[Description]:
BET bromodomain inhibitor is a potent BET inhibitor extracted from patent WO/2015/153871A2, compound example 11.
[Related Catalog]:
[Target]
BET[1]
[References]
[1]. WO/2015/153871A2
[Related Small Molecules]
(+)-JQ1
|
GSK126
|
Tazemetostat (EPZ-6438)
|
Birabresib (OTX015)
|
A 485
|
Curcumin
|
ARV-771
|
ARV-825
|
I-BET762
|
BI 2536
|
GSK343
|
C646
|
3-Deazaneplanocin A (hydrochloride)
|
I-BET151
|
666-15
Chemical & Physical Properties
[ Molecular Formula ]:
C24H20ClN5O2
[ Molecular Weight ]:
445.90100
[ Exact Mass ]:
445.13100
[ PSA ]:
99.30000
[ LogP ]:
4.60730
[ Storage condition ]:
2-8℃