S07-2009

Names

[ CAS No. ]:
1580241-55-9

[ Name ]:
S07-2009

Biological Activity

[Description]:

S07-2009 is a potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitor with an IC50 value of 0.20 μM[1].

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> Others >> Others

[Target]

IC50: 0.20 ± 0.12 μM (AKR1C3), 11.18 ± 4.39 μM (AKR1C1), 5.71 ± 2.78 μM (AKR1C2)[1]

[References]

[1]. Siyu He, et al. Discovery of Novel Aldo-Keto Reductase 1C3 Inhibitors as Chemotherapeutic Potentiators for Cancer Drug Resistance. ACS Med. Chem. Lett. Jun 2022.

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₆H₁₉N₃O₅

[ Molecular Weight ]:
333.34

Related Compounds