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GSK121 (trifluoroacetate salt)

Names

[ CAS No. ]:
1652591-80-4

[ Name ]:
GSK121 (trifluoroacetate salt)

[Synonym ]:
(3-Amino-1-piperidinyl)[1-methyl-2-(1-methyl-1H-indol-2-yl)-1H-benzimidazol-5-yl]methanone trifluoroacetate (1:1)
(3-Aminopiperidin-1-yl)(1-methyl-2-(1-methyl-1H-indol-2-yl)-1H-benzo[d]imidazol-5-yl)methanone trifluoroacetic acid salt
Acetic acid, 2,2,2-trifluoro-, compd. with (3-amino-1-piperidinyl)[1-methyl-2-(1-methyl-1H-indol-2-yl)-1H-benzimidazol-5-yl]methanone (1:1)
GSK121 (trifluoroacetate salt)

Biological Activity

[Description]:

GSK-121 Trifluoroacetates a selective PAD4 inhibitor[1].

[Related Catalog]:

Research Areas >> Cancer
Research Areas >> Cardiovascular Disease
Research Areas >> Inflammation/Immunology
Signaling Pathways >> Epigenetics >> Protein Arginine Deiminase

[References]

[1]. Drewes G, et al. Inhibition of PAD4 activity is sufficient to disrupt mouse and human NET formation. Nat Chem Biol. 2015 Mar;11(3):189-91.

Chemical & Physical Properties

[ Molecular Formula ]:
C25H26F3N5O3

[ Molecular Weight ]:
501.501

[ Exact Mass ]:
501.198761

Related Compounds