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BET-IN-4

Names

[ CAS No. ]:
1801503-93-4

[ Name ]:
BET-IN-4

Biological Activity

[Description]:

BET-IN-4 is a potent BET bromodomain protein (BRD4) inhibitor, with an IC50 of ≤ 1 μM[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain

[Target]

BRD4:≤ 1 μM (IC50)


[In Vitro]

BET-IN-4 (Compound 50) is a potent BET bromodomain protein (BRD4) inhibitor, with an IC50 of ≤ 1 μM[1].

[References]

[1]. Susanta Samajdar, et al. Bicyclic heterocyclic derivatives as bromodomain inhibitors. WO2015104653A1

Chemical & Physical Properties

[ Molecular Formula ]:
C22H21N3O3

[ Molecular Weight ]:
375.42


Related Compounds