BRD-IN-26

Names

[ CAS No. ]:
1915012-19-9

[ Name ]:
BRD-IN-26

Biological Activity

[Description]:

BRD-IN-26 is a potent bromodomain inhibitor that binds the fifth bromodomain of PB1 with a KD of 124 nM, SMARCA2B and SMARCA4 with KD values of 262 and 417 nM, respectively; displays excellent selectivity over other bromodomains.

[References]

References 1. Sutherell CL, et al. J Med Chem. 2016 May 26;59(10):5095-101. View Related Products by Target Bromodomain

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₇H₁₉ClN₄O

[ Molecular Weight ]:
330.816

Related Compounds

brd-in-3
BRD-IN-17
EGFR-IN-26
HDAC-IN-26
PI3K-IN-26
HPK1-IN-26
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