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PROTAC BET Degrader-10

Names

[ CAS No. ]:
1957234-97-7

[ Name ]:
PROTAC BET Degrader-10

Biological Activity

[Description]:

PROTAC BET Degrader-10 is a potent BET protein BRD4 degrader extracted from patent WO2017007612A1, example 37, with a DC50 of 49 nM[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> PROTAC >> PROTAC
Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain

[References]

[1]. James Bradner, et al. Methods to induce targeted protein degradation through bifunctional molecules. WO2017007612A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C39H39ClN8O6S

[ Molecular Weight ]:
783.29

[ Storage condition ]:
-20°C

Related Compounds