CCG 224061
Names
[ CAS No. ]:
2055990-82-2
[ Name ]:
CCG 224061
Biological Activity
[Description]:
A potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 66 nM; displays >30-fold selectivity over GRK5, GRK1, PKA and ROCK1.
[References]
References 1. Bouley R, et al. Mol Pharmacol. 2017 Dec;92(6):707-717. View Related Products by Target GRK (GPCRK)
Chemical & Physical Properties
[ Molecular Formula ]:
C19H20FN3O
[ Molecular Weight ]:
325.387