BCL6 inhibitor 7

Names

[ CAS No. ]:
2097518-46-0

[ Name ]:
BCL6 inhibitor 7

Biological Activity

[Description]:

A potent BCL6 protein-protein interaction inhibitor with Kd of 78 nM; exhibits an efficacy in cell-free and cellular PPI assays (ELISA IC50= 480 nM, M2H IC50= 8.6 uM).

[References]

References 1. Kamada Y, et al. J Med Chem. 2017 May 25;60(10):4358-4368. View Related Products by Target Bcl-2

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₈H₁₅ClN₆O

[ Molecular Weight ]:
366.809

Related Compounds

BCL6 inhibitor 8c
ATX inhibitor 7
Tubulin inhibitor 7
KRAS inhibitor-7
Microtubule inhibitor 7
Thrombin inhibitor 7
1-Nitroso-2-phenylazepane
4-((Cyclohexylamino)methyl)benzoic acid hydrochloride
6-(1-Benzyl-1h-pyrazol-5-yl)-1-cyclopentyl-3-ethyl-1h-indazole
4,5-Dihydro-3-(4-nitrophenyl)isoxazole
(Z)-4-methoxy-2,3-dimethyl-4-oxobut-2-enoic acid
1-[(2,4-Dichlorophenyl)methyl]-N-(1,1-dimethylethyl)-2-methyl-1H-indole-3-methanamine
N-(2-cyclopropanecarbonyl-1,2,3,4-tetrahydroisoquinolin-7-yl)adamantane-1-carboxamide
N-[1-(4-fluorophenyl)-5-oxopyrrolidin-3-yl]-4-hydroxypiperidine-1-carboxamide
2-Methoxy-6-(pyrazol-1-yl)-benzonitrile
1H-3-Benzazepin-7-ol, 8-chloro-2,3,4,5-tetrahydro-5-(3-iodophenyl)-3-methyl-, (S)-