TRV0109101 hydrochloride
Names
[ CAS No. ]:
2101210-22-2
[ Name ]:
TRV0109101 hydrochloride
[Synonym ]:
6-Oxaspiro[4.5]decane-9-ethanamine, 9-(2-pyridinyl)-N-(2-thienylmethyl)-, (9R)-, hydrochloride (1:1)
2-[(9R)-9-(2-Pyridinyl)-6-oxaspiro[4.5]dec-9-yl]-N-(2-thienylmethyl)ethanamine hydrochloride (1:1)
Biological Activity
[Description]:
A selective, G protein-biased µ-opioid receptor agonist, does not promote the development of opioid-induced mechanical allodynia (OIMA) and rapidly reverses allodynia in vivo.
[References]
References 1. Koblish M, et al. J Pharmacol Exp Ther. 2017 Aug;362(2):254-262. View Related Products by Target Opioid Receptor
Chemical & Physical Properties
[ Molecular Formula ]:
C21H29ClN2OS
[ Molecular Weight ]:
392.986
[ Exact Mass ]:
392.168915