(S,R,S)-AHPC-amido-C5-acid

Names

[ Name ]:
(S,R,S)-AHPC-amido-C5-acid

Biological Activity

[Description]:

(S,R,S)-AHPC-amido-C5-acid incorporates a VHL ligand for the E3 ubiquitin ligase, and a PROTAC linker. (S,R,S)-AHPC-amido-C5-acid can be used to design XY028-133 (HY-129180)[1].

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> PROTAC >> PROTAC Linker

[References]

[1]. Jian Jin, et al. Compositions and methods for treating cdk4/6-mediated cancer. WO2018106870A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₉H₄₀N₄O₆S

[ Molecular Weight ]:
572.72

(S,R,S)-AHPC-amido-C5-acid

Names

Biological Activity

Chemical & Physical Properties

Related Compounds