CARM1 inhibitor 9
Names
[ CAS No. ]:
2180931-09-1
[ Name ]:
CARM1 inhibitor 9
Biological Activity
[Description]:
CARM1 inhibitor 9 is a potent, selective inhibitor of arginine methyltransferase 1 (CARM1, PRMT4) with IC50 of 94 nM; displays 20-fold selective for CARM1 over PRMT6 and highly selective over PRMT1, PRMT3, PRMT8 as well as PRMT5 and PRMT7; CARM1 inhibitor 9 is a useful tool for studying the role of CARM1 in health and disease.
[References]
References 1. Kaniskan HÜ, et al. Medchemcomm. 2016 Sep 1;7(9):1793-1796. View Related Products by Target Histone Methyltransferase (HMTase)
Chemical & Physical Properties
[ Molecular Formula ]:
C15H24BrN3
[ Molecular Weight ]:
326.282