PROTAC ERRα Degrader-2

Names

[ Name ]:
PROTAC ERRα Degrader-2

Biological Activity

[Description]:

PROTAC ERRalpha Degrader-2 comprises a MDM2 ligand binding group, a linker and an estrogen-related receptor alpha (ERRa) binding group. PROTAC ERRalpha Degrader-2 is an estrogen-related receptor alpha (ERRa) degrader[1].

[Related Catalog]:

Signaling Pathways >> Others >> Estrogen Receptor/ERR

Research Areas >> Cancer

Signaling Pathways >> PROTAC >> PROTAC

[References]

[1]. Peng L, et al. Identification of New Small-Molecule Inducers of Estrogen-related Receptor α (ERRα) Degradation. ACS Med Chem Lett. 2019 Apr 12;10(5):767-772.

Chemical & Physical Properties

[ Molecular Formula ]:
C₅₇H₅₅Cl₂F₆N₇O₈

[ Molecular Weight ]:
1150.99

[ Storage condition ]:
2-8°C