TEAD-IN-3

Names

[ Name ]:
TEAD-IN-3

Biological Activity

[Description]:

TEAD-IN-3 (compound I-177) is a potent TEAD transcription factor inhibitor. TEAD-IN-3 can be used for the research of proliferative diseases (such as cancer) [1].

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> Stem Cell/Wnt >> YAP

[References]

[1]. Nathanael S. Gray, et al. Transcriptional enhanced associate domain (tead) transcription factor inhibitors and uses thereof. WO2020081572A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₂H₂₀F₃N₅O₂

[ Molecular Weight ]:
443.42

Related Compounds

TEAD-IN-2
TEAD-IN-2
DUBs-IN-3
CETP-IN-3
ILK-IN-3
CD80-IN-3
4-((Cyclohexylamino)methyl)benzoic acid hydrochloride
1-[(2,4-Dichlorophenyl)methyl]-N-(1,1-dimethylethyl)-2-methyl-1H-indole-3-methanamine
2-Methoxy-6-(pyrazol-1-yl)-benzonitrile
1H-3-Benzazepin-7-ol, 8-chloro-2,3,4,5-tetrahydro-5-(3-iodophenyl)-3-methyl-, (S)-
(4-Methyl-tetrahydro-furan-2-yl)-methanol
N-(1-cyanocyclopentyl)-2-[4-(4-fluorobenzenesulfonyl)-1,4-diazepan-1-yl]acetamide
4,5,6,7-Tetrahydrobenzo[d]isoxazole-3-carbaldehyde
tert-Butyl-DL-alanine
4-amino-N-[2-tert-butyl-1-(tetrahydro-2H-pyran-4-ylmethyl)-1H-benzimidazol-5-yl]-N-ethylbenzenesulfonamide
3-Furancarboxylic acid, 4-amino-2,5-dihydro-5-oxo-, ethyl ester