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GRK2 Inhibitor

Names

[ CAS No. ]:
24269-96-3

[ Name ]:
GRK2 Inhibitor

[Synonym ]:
5-[2-(5-nitro-furan-2-yl)-vinyl]-furan-2-carboxylic acid methyl ester
5-[2-(5-Nitro-2-furanyl)ethenyl]-2-furancarboxylic Acid Methyl Ester

Biological Activity

[Description]:

GRK2 Inhibitor 1 (methyl 5-[2-(5-nitro-2-furyl)vinyl]-2-furoate) is a GRK2 (β-ARK1) inhibitor[1].

[Related Catalog]:

Research Areas >> Cardiovascular Disease
Signaling Pathways >> Others >> Others

[References]

[1]. Nimitvilai S, et al. Reversal of dopamine D2 agonist-induced inhibition of ventral tegmental area neurons by Gq-linked neurotransmitters is dependent on protein kinase C, G protein-coupled receptor kinase, and dynamin. J Pharmacol Exp Ther. 2013 Jan;344(1):253-63.

Chemical & Physical Properties

[ Molecular Formula ]:
C12H9NO6

[ Molecular Weight ]:
263.20

[ Exact Mass ]:
263.04300

[ PSA ]:
98.40000

[ LogP ]:
3.26100

Related Compounds