Palosuran hydrochloride
Names
[ CAS No. ]:
2469274-58-4
[ Name ]:
Palosuran hydrochloride
Biological Activity
[Description]:
Palosuran hydrochloride (ACT-058362 hydrochloride) is a potent, selective, and orally active antagonist of urotensin II receptor, with an IC50 of 3.6 nM for CHO cell membranes expressing human recombinant receptors. Palosuran hydrochloride can improves pancreatic and renal function in diabetic rats.
Chemical & Physical Properties
[ Molecular Formula ]:
C25H31ClN4O2
[ Molecular Weight ]:
454.99