<Suppliers Price>

PROTAC ERα Y537S degrader-1

Names

[ CAS No. ]:
2667598-05-0

[ Name ]:
PROTAC ERα Y537S degrader-1

Biological Activity

[Description]:

PROTAC ERα Y537S degrader-1 comprises a ubiquitin E3 ligase binding group, a linker and a protein binding group. PROTAC ERα Y537S degrader-1 extracts from patent WO2021143822, example 12. PROTAC ERα Y537S degrader-1 is an estrogen receptor-alpha (ERα) Y537S degrader[1].

[Related Catalog]:

Signaling Pathways >> Others >> Estrogen Receptor/ERR
Research Areas >> Cancer
Signaling Pathways >> PROTAC >> PROTAC

[References]

[1]. Yang FL, et, al. Bicyclic imide derivative, preparation method thereof, and application thereof in medicine. WO2021143822A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C46H49N5O6

[ Molecular Weight ]:
767.91


Related Compounds