BRD4-BD1/2-IN-2

Names

[ Name ]:
BRD4-BD1/2-IN-2

Biological Activity

[Description]:

BRD4-BD1/2-IN-2 is a potent BRD4 BD2 inhibitor with IC50s of <0.5 nM and <300 nM for BRD4 BD2 and BRD4 BD1, respectively (WO2021233371A1, compound 2)[1].

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain

[References]

[1]. Compound functioning as bromodomain protein inhibitor, and composition. WO2021233371A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C₃₀H₃₃N₅O₄

[ Molecular Weight ]:
527.61

BRD4-BD1/2-IN-2

Names

Biological Activity

Chemical & Physical Properties

Related Compounds