BRD4 Inhibitor-23

Names

[ CAS No. ]:
2760307-53-5

[ Name ]:
BRD4 Inhibitor-23

Biological Activity

[Description]:

BRD4 Inhibitor-23 is a potent and orally active BRD4 inhibitor with IC50s of 6.21 nM and 1.44 nM for BRD4 BD-1 and BRD4 BD-2, respectively (WO2022033542A1; Example 1)[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain

[References]

[1]. Chunli Shen, et al. 5-membered heteroaromatic pyridone compounds and application thereof. WO2022033542A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C22H19F2N3O4S

[ Molecular Weight ]:
459.47

Related Compounds