Org 42599
Names
[ CAS No. ]:
501444-89-9
[ Name ]:
Org 42599
Biological Activity
[Description]:
Org 42599 is a cell-permeant, allosterically binding, small-molecule agonist of luteinizing hormone (LH) receptor that rescues the folding and cell surface expression mutant mutant human LH receptors A593P and S616Y (EC50=70.8 nM).
[References]
References 1. Newton CL, et al. Proc Natl Acad Sci U S A. 2011 Apr 26;108(17):7172-6. View Related Products by Target Luteinizing Hormone Receptor (LHR)
Chemical & Physical Properties
[ Molecular Formula ]:
C26H31F3N6O5S2
[ Molecular Weight ]:
628.686