Carprazidil

Names

[ Name ]:
Carprazidil

[Synonym ]:
Carprazidil
Carprazidilum
Carprazidilum [INN-Latin]
methyl 2-oxo-5-(1,2,3,6-tetrahydro-1-pyridyl)-2,8-dihydro<1,2,4>oxadiazolo<2,3-a>pyrimidine-7-carbamate
Carprazadil
Carprazidilo
Methyl 5-(3,6-dihydro-1(2H)-pyridyl)-2-oxo-2H-(1,2,4)oxadiazolo(2,3-a)pyrimidine-7-carbamate

Biological Activity

[Description]:

Carprazidil is a potent vasodilator used to treat severe hypertension and mild heart failure.

[References]

1. Bianchetti MG, et al. Comparative evaluation of the new vasodilator carprazidil and minoxidil in the treatment of moderate to severe hypertension. Eur J Clin Pharmacol. 1982;23(6):483-9.

Chemical & Physical Properties

[ Density]:
1.59g/cm3

[ Molecular Formula ]:
C₁₂H₁₃N₅O₄

[ Molecular Weight ]:
291.26300

[ Exact Mass ]:
291.09700

[ PSA ]:
101.97000

[ LogP ]:
0.76510

[ Index of Refraction ]:
1.712

Carprazidil

Names

Biological Activity

Chemical & Physical Properties

Synthetic Route

Click to get detail synthetic route

Precursor & DownStream

Precursor

DownStream

Related Compounds