Tec Kinase-IN-6

Names

[ Name ]:
Tec Kinase-IN-6

Biological Activity

[Description]:

A selecitve small molecule toward Tec kinase-mediated tyrosine phosphorylation of FGF2 with IC50 of 8.9 uM; inhibits Tec-FGF2 complex and blocks tyrosine phosphorylation of FGF2 in cells, also inhibit FGF2 secretion from cells.

[References]

References 1. La Venuta G, et al. J Biol Chem. 2016 Aug 19;291(34):17787-803. View Related Products by Target Tec Kinase

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₉H₁₉N₃O₅

[ Molecular Weight ]:
369.377

Related Compounds

Tec Kinase-IN-21
Tec Kinase-IN-14
IRE1α kinase-IN-6
MET kinase-IN-2
Multi-kinase-IN-1
IRE1α kinase-IN-3
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