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PAR-2 (6-1) amide (human) trifluoroacetate salt

Names

[ CAS No. ]:
942413-05-0

[ Name ]:
PAR-2 (6-1) amide (human) trifluoroacetate salt

Biological Activity

[Description]:

VKGILS-NH2 is a reversed amino acid sequence control peptide for SLIGKV-NH2 (protease-activated receptor 2 (PAR2) agonist). VKGILS-NH2 has no effect on DNA synthesis in cells[1][2].

[Related Catalog]:

Signaling Pathways >> Others >> Others
Research Areas >> Inflammation/Immunology

[References]

[1]. M Tognetto, et al. Evidence That PAR-1 and PAR-2 Mediate Prostanoid-Dependent Contraction in Isolated Guinea-Pig Gallbladder. Br J Pharmacol. 2000 Oct;131(4):689-94.

[2]. David A Vesey, et al. Proinflammatory and Proliferative Responses of Human Proximal Tubule Cells to PAR-2 Activation. Am J Physiol Renal Physiol. 2007 Nov;293(5):F1441-9.

Chemical & Physical Properties

[ Molecular Formula ]:
C28H54N8O7

[ Molecular Weight ]:
614.77800

[ Exact Mass ]:
614.41200

[ PSA ]:
260.86000

[ LogP ]:
1.77930

Related Compounds