870812-93-4

• 常用中文名：N-苄氧羰基-4-[(3R)-3-氨基-1-氧-4-(苯硫基)丁基]吗啉
• 常用英文名：N-Benzyloxycarbonyl-4-[(3R)-3-amino-1-oxo-4-(phenylthio)butyl]morpholine
• CAS号：870812-93-4
• 分子式：C₂₂H₂₆N₂O₄S
• 分子量：414.51800
• 发布时间：2018-07-31 18:21:10
• 更新时间：2024-01-31 20:11:42

名称

• 中文名: (1R)-3-(4-吗啉)-3-氧代-1-((苯基磺酰基)甲基)丙基氨基甲酸苄酯
• 英文名: benzyl N-[(2R)-4-morpholin-4-yl-4-oxo-1-phenylsulfanylbutan-2-yl]carbamate
• 英文别名: (R)-benzyl 4-morpholino-4-oxo-1-(phenylthio)butan-2-ylcarbamate; N-Benzyloxycarbonyl-4-[(3R)-3-amino-1-oxo-4-(phenylthio)butyl]morpholine; N-[(1R)-3-(4-Morpholinyl)-3-oxo-1-[(phenylthio)methyl]propyl]carbamic Acid Phenylmethyl Ester; benzyl (1R)-3-(4-morpholinyl)-3-oxo-1-((phenylsulfanyl)methyl)propylcarbamate; [(1R)-3-(4-Morpholinyl)-3-oxo-1-[(phenylthio)methyl]propyl]carbamic Acid Benzyl Ester

物化性质

• 分子式: C₂₂H₂₆N₂O₄S
• 分子量: 414.51800
• 精确质量: 414.16100
• PSA: 96.66000
• LogP: 3.46490

合成路线

870812-92-3 882-33-7 ~74% 870812-93-4

文献：Elmore, Steven W.; Bruncko, Milan; Park, Cheol-Min Patent: US2005/272744 A1, 2005 ; Location in patent: Page/Page column 20 ; US 20050272744 A1

1027345-09-0 108-98-5 ~46% 870812-93-4

文献：GENENTECH, INC.; WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH Patent: WO2008/61208 A2, 2008 ; Location in patent: Page/Page column 31; 33 ; WO 2008/061208 A2

75443-62-8 ~% 870812-93-4

文献：ASTRAZENECA AB Patent: US2012/35134 A1, 2012 ;

118399-28-3 ~% 870812-93-4

文献：ASTRAZENECA AB Patent: US2012/35134 A1, 2012 ;

123673-31-4 ~% 870812-93-4

文献：ASTRAZENECA AB Patent: US2012/35134 A1, 2012 ;

78663-07-7 ~% 870812-93-4

文献：ASTRAZENECA AB Patent: US2012/35134 A1, 2012 ;

上下游产品

上游产品  6
870812-92-3 882-33-7 108-98-5 75443-62-8
118399-28-3 78663-07-7
下游产品  1
870812-94-5