PF-06459988
Names
[ CAS No. ]:
1428774-45-1
[ Name ]:
PF-06459988
[Synonym ]:
1-((3R,4R)-3-(((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)oxy)methyl)-4-methoxypyrrolidin-1-yl)prop-2-en-1-one
Biological Activity
[Description]:
PF-06459988 is an irreversible inhibitor of T790M-Containing EGFR Mutants.
[Related Catalog]:
[Target]
IC50: 45 nM (H1975 EGFR), 3.3 μM (EGFR)
[References]
[Related Small Molecules]
Chemical & Physical Properties
[ Storage condition ]:
2-8℃
Safety Information
[ RIDADR ]:
NONH for all modes of transport