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Mal-C6-α-Amanitin

Names

[ CAS No. ]:
1578249-76-9

[ Name ]:
Mal-C6-α-Amanitin

Biological Activity

[Description]:

Mal-C6-α-Amanitin is a drug-linker conjugate for ADC with potent antitumor activity by using α-Amanitin (an RNA polymerase II inhibitor), linked via the ADC linker Mal-C6.

[Related Catalog]:

Research Areas >> Cancer

[Target]

Daunorubicins/Doxorubicins


[References]

[1]. Brian Lannutti,et al. Ror1 antibody immunoconjugates. WO2018237335A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C55H78N12O17S

[ Molecular Weight ]:
1211.34


Related Compounds