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GP3269

Names

[ CAS No. ]:
186393-42-0

[ Name ]:
GP3269

Biological Activity

[Description]:

GP3269 is a potent, selective, and orally active inhibitor of human adenosine kinase (AK) with an IC50 of 11 nM. GP3269 exhibits anticonvulsant activity in rats[1].

[Related Catalog]:

Signaling Pathways >> Neuronal Signaling >> Adenosine Kinase
Research Areas >> Neurological Disease
Signaling Pathways >> Metabolic Enzyme/Protease >> Adenosine Kinase

[References]

[1]. Mark D. ErionGensia, et al. Design, Synthesis and Anticonvulsant Activity of the Potent Adenosine Kinase Inhibitor GP3269.

Chemical & Physical Properties

[ Molecular Formula ]:
C23H21FN4O3

[ Molecular Weight ]:
420.44

Related Compounds