LKY-047
Names
[ CAS No. ]:
1954681-29-8
[ Name ]:
LKY-047
Biological Activity
[Description]:
LKY-047, a Decursin derivative, is a potent and selective reversible competitive cytochrome P45022J2 (CYP2J2) inhibitor with an IC50 of 1.7 μM. LKY-047 is inactive against other human P450s, such as CYPs 1A2, 2A6, 2B6, 2C8, 2C9, 2C19, 2D6, 2E1, and 3A.
Chemical & Physical Properties
[ Molecular Formula ]:
C23H19NO7
[ Molecular Weight ]:
421.40