PI3Kδ-IN-8
Names
[ CAS No. ]:
2101518-75-4
[ Name ]:
PI3Kδ-IN-8
Biological Activity
[Description]:
PI3Kδ-IN-8 is a potent, selective and orally active PI3Kδ, with an IC50 of 3.3 nM. PI3Kδ-IN-8 shows selectivity for PI3Kδ over PI3Kα, PI3Kβ, and PI3Kγ (IC50=377.2, 241.6, 17.9 nM, respectively). PI3Kδ-IN-8 has anti-tumor activity.
Chemical & Physical Properties
[ Molecular Formula ]:
C28H21F2N7O
[ Molecular Weight ]:
509.51