LSD1-IN-11p
Names
[ CAS No. ]:
2101951-67-9
[ Name ]:
LSD1-IN-11p
Biological Activity
[Description]:
LSD1-IN-11p is a reversible LSD1 inhibitor with IC50/Kd of 79/21 nM; upregulates the expression of the surrogate cellular biomarker CD86 (IC50=0.52 uM); has moderate oral bioavailability in mice (F%=38%).
[References]
References 1. Mould DP, et al. Bioorg Med Chem Lett. 2017 Jul 15;27(14):3190-3195. View Related Products by Target Histone Demethylase
Chemical & Physical Properties
[ Molecular Formula ]:
C22H24N6O3
[ Molecular Weight ]:
420.473