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BLU-782

Names

[ CAS No. ]:
2141955-96-4

[ Name ]:
BLU-782

Biological Activity

[Description]:

ALK2-IN-1 is a activin receptor-like kinase-2 (ALK2) inhibitor extracted from patent WO2017181117A1, Compound 876, has an IC50 of <10 nM[1].

[Related Catalog]:

Research Areas >> Cancer

[Target]

IC50: <10 nM (ALK2)[1]


[References]

[1]. Natasja Brooijmans, et al. Inhibitors of activin receptor-like kinase. WO2017181117A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C31H42N6O4

[ Molecular Weight ]:
562.70


Related Compounds