TT-10
Names
[ CAS No. ]:
2230640-94-3
[ Name ]:
TT-10
Biological Activity
[Description]:
TT-10 (YAP-TEAD activator TT-10) is a small molecule activator that activates pro-proliferative YES-associated protein (YAP) and transcriptional enhancer factor domain (TEAD) activities in cardiomyocytes; promoted cardiomyocyte proliferation and simultaneously exerted antioxidant and antiapoptotic effects in vitro via nuclear translocation of YAP, activates YAP-TEADs activity and the Wnt/β-Catenin signaling pathway; ameliorates cardiac dysfunction, decreases ROS and DNA aamage and apoptosis after myocardial infarction (MI) in mice.
[References]
References 1. Hara H, et al. JACC Basic Transl Sci. 2018 Nov 12;3(5):639-653. View Related Products by Target Yes-associated Protein (YAP)
Chemical & Physical Properties
[ Molecular Formula ]:
C11H10FN3OS2
[ Molecular Weight ]:
283.339