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PKC-IN-7

Names

[ CAS No. ]:
860468-10-6

[ Name ]:
PKC-IN-7

Biological Activity

[Description]:

PKC-IN-7 is a potent, selective, reversible, ATP-competitive PKCα/β inhibitor with IC50 of 4.7/3.3 nM; dispalys >50-fold selectivity against PKC isotypes δ,ε,η,θ and other kinases belonging to the AGC family; inhibits IgM-stimulated mouse B cell proliferation with an IC50 of 296 nM.

[References]

References 1. van Eis MJ, et al. Bioorg Med Chem Lett. 2017 Feb 15;27(4):781-786. View Related Products by Target PKC

Chemical & Physical Properties

[ Molecular Formula ]:
C26H22ClN3O2

[ Molecular Weight ]:
443.931


Related Compounds