N-butyl-4-methoxy-7,7-dimethyl-6,8-dihydropyrimido[4,5-b][1,4]benzothiazin-9-amine,hydrobromide

Names

[ CAS No. ]:
102688-85-7

[ Name ]:
N-butyl-4-methoxy-7,7-dimethyl-6,8-dihydropyrimido[4,5-b][1,4]benzothiazin-9-amine,hydrobromide

[Synonym ]:
N-butyl-4-methoxy-7,7-dimethyl-6,8-dihydropyrimido[4,5-b][1,4]benzothiazin-9-amine
4-Methoxy-7,7-dimethyl-9-butylamino-7,8-dihydro-1,3-diazaphenothiazine hydrobromide
6H-Pyrimido(4,5-b)(1,4)benzothiazin-9-amine,7,8-dihydro-N-butyl-7,7-dimethyl-4-methoxy-,monohydrobromide
7,8-Dihydro-N-butyl-7,7-dimethyl-4-methoxy-6H-pyrimido(4,5-b)(1,4)benzothiazin-9-amine HBr

Chemical & Physical Properties

[ Molecular Formula ]:
C17H25BrN4OS

[ Molecular Weight ]:
413.37600

[ Exact Mass ]:
412.09300

[ PSA ]:
84.70000

[ LogP ]:
4.86930

Toxicological Information

CHEMICAL IDENTIFICATION

RTECS NUMBER :
UW7681515
CHEMICAL NAME :
6H-Pyrimido(4,5-b)(1,4)benzothiazin-9-amine, 7,8-dihydro-N-butyl-7,7-dimethyl-4-methoxy-, monohydrobromide
CAS REGISTRY NUMBER :
102688-85-7
LAST UPDATED :
198906
DATA ITEMS CITED :
1
MOLECULAR FORMULA :
C17-H24-N4-O-S.Br-H
MOLECULAR WEIGHT :
413.43

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Unreported
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
255 mg/kg
TOXIC EFFECTS :
Behavioral - altered sleep time (including change in righting reflex) Behavioral - convulsions or effect on seizure threshold Behavioral - changes in motor activity (specific assay)
REFERENCE :
PCJOAU Pharmaceutical Chemistry Journal (English Translation). Translation of KHFZAN. (Plenum Pub. Corp., 233 Spring St., New York, NY 10013) No.1- 1967- Volume(issue)/page/year: 19,459,1985

Related Compounds