Rac-PQ-912
Names
[ CAS No. ]:
1276021-63-6
[ Name ]:
Rac-PQ-912
Biological Activity
[Description]:
Rac-PQ-912 is a glutaminyl cyclase (QC) inhibitor extracted from patent WO2011029920A1, compound example 12, has an EC50 of 482 nM and a Ki of 62.5 nM for hQC[1].
[Related Catalog]:
[Target]
EC50: 482 nM (hQC) Ki: 62.5 nM (hQC)[1]
[References]
Chemical & Physical Properties
[ Molecular Formula ]:
C19H20N4O2
[ Molecular Weight ]:
336.39