4-amino-8-fluoro-N-(2-pyrrolidin-1-ylethyl)cinnoline-3-carboxamide

Names

[ CAS No. ]:
187231-62-5

[ Name ]:
4-amino-8-fluoro-N-(2-pyrrolidin-1-ylethyl)cinnoline-3-carboxamide

[Synonym ]:
4-AMINO-8-FLUORO-N-(2-(PYRROLIDIN-1-YL)ETHYL)-3-CINNOLINECARBOXAMIDE
4-Amino-8-fluoro-N-(2-(1-pyrrolidinyl)ethyl)-3-cinnolinecarboxamide
3-Cinnolinecarboxamide,4-amino-8-fluoro-N-(2-(1-pyrrolidinyl)ethyl)

Chemical & Physical Properties

[ Density]:
1.323g/cm3

[ Boiling Point ]:
425.5ºC at 760 mmHg

[ Molecular Formula ]:
C15H18FN5O

[ Molecular Weight ]:
303.33500

[ Flash Point ]:
211.1ºC

[ Exact Mass ]:
303.15000

[ PSA ]:
84.14000

[ LogP ]:
2.08670

[ Vapour Pressure ]:
1.91E-07mmHg at 25°C

[ Index of Refraction ]:
1.642

Toxicological Information

CHEMICAL IDENTIFICATION

RTECS NUMBER :
GE3620942
CHEMICAL NAME :
3-Cinnolinecarboxamide, 4-amino-8-fluoro-N-(2-(1-pyrrolidinyl)ethyl)-
CAS REGISTRY NUMBER :
187231-62-5
LAST UPDATED :
199803
DATA ITEMS CITED :
2
MOLECULAR FORMULA :
C15-H18-F-N5-O
MOLECULAR WEIGHT :
303.38

HEALTH HAZARD DATA

ACUTE TOXICITY DATA

TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Oral
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
1250 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
PHARAT Pharmazie. (VEB Verlag Volk und Gesundheit, Neue Gruenstr. 18, Berlin DDR-1020, Ger. Dem. Rep.) V.1- 1946- Volume(issue)/page/year: 52,91,1997
TYPE OF TEST :
LD50 - Lethal dose, 50 percent kill
ROUTE OF EXPOSURE :
Intraperitoneal
SPECIES OBSERVED :
Rodent - mouse
DOSE/DURATION :
750 mg/kg
TOXIC EFFECTS :
Details of toxic effects not reported other than lethal dose value
REFERENCE :
PHARAT Pharmazie. (VEB Verlag Volk und Gesundheit, Neue Gruenstr. 18, Berlin DDR-1020, Ger. Dem. Rep.) V.1- 1946- Volume(issue)/page/year: 52,91,1997

Related Compounds