p38α inhibitor 2
Modify Date: 2024-01-22 13:53:26
p38α inhibitor 2 structure
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Common Name | p38α inhibitor 2 | ||
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| CAS Number | 1095003-80-7 | Molecular Weight | 475.58 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C27H33N5O3 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of p38α inhibitor 2p38α inhibitor 2 is a highly potent and selective p38α MAPK inhibitor, with a pIC50 of 9.6. p38α inhibitor 2 inhibits the hERG ion channel (IC50=27 μM) and shows a promising selectivity profile when tested in a panel of 51 other protein kinases (<30% inhibition at 10 μM concentration) and a panel of 141 other biological targets. |
| Name | p38α inhibitor 2 |
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| Description | p38α inhibitor 2 is a highly potent and selective p38α MAPK inhibitor, with a pIC50 of 9.6. p38α inhibitor 2 inhibits the hERG ion channel (IC50=27 μM) and shows a promising selectivity profile when tested in a panel of 51 other protein kinases (<30% inhibition at 10 μM concentration) and a panel of 141 other biological targets. |
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| Molecular Formula | C27H33N5O3 |
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| Molecular Weight | 475.58 |