Eletriptan-d5
Modify Date: 2024-01-06 12:17:56
Eletriptan-d5 structure
|
Common Name | Eletriptan-d5 | ||
|---|---|---|---|---|
| CAS Number | 1126745-65-0 | Molecular Weight | 387.55000 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C22H21D5N2O2S | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of Eletriptan-d5Eletriptan-d5 is the deuterium labeled Eletriptan[1]. Eletriptan (UK-116044) is a highly selective and orally active serotonin 5-HT1B and 5-HT1D receptor agonist, with pKi values of 8.0 and 8.9, respectively. Eletriptan has inhibitory effects on markers of neurogenic inflammation in rats. Eletriptan can be used for researching migraine[2]. |
| Name | Eletriptan-d5 |
|---|---|
| Synonym | More Synonyms |
| Description | Eletriptan-d5 is the deuterium labeled Eletriptan[1]. Eletriptan (UK-116044) is a highly selective and orally active serotonin 5-HT1B and 5-HT1D receptor agonist, with pKi values of 8.0 and 8.9, respectively. Eletriptan has inhibitory effects on markers of neurogenic inflammation in rats. Eletriptan can be used for researching migraine[2]. |
|---|---|
| Related Catalog | |
| In Vitro | Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1]. |
| References |
| Molecular Formula | C22H21D5N2O2S |
|---|---|
| Molecular Weight | 387.55000 |
| Exact Mass | 387.20300 |
| PSA | 61.55000 |
| LogP | 4.83970 |
| Eletriptan-d5 |