Ralaniten acetate

Modify Date: 2022-01-29 14:27:10

Ralaniten acetate Structure
Ralaniten acetate structure
Common Name Ralaniten acetate
CAS Number 1637573-02-4 Molecular Weight 436.929
Density N/A Boiling Point N/A
Molecular Formula C23H29ClO6 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Ralaniten acetate


A novel small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor for the treatment of advanced prostate cancer; AR NTD-targeting agents have the potential to overcome shortcomings of current hormonal therapies by inhibiting all forms of AR-mediated transcriptional activity, and as a result, may affect a broader AR population including mutational and splice variant ARs. Prostate Cancer Phase 2 Clinical

 Names

Name Ralaniten acetate

 Ralaniten acetate Biological Activity

Description A novel small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor for the treatment of advanced prostate cancer; AR NTD-targeting agents have the potential to overcome shortcomings of current hormonal therapies by inhibiting all forms of AR-mediated transcriptional activity, and as a result, may affect a broader AR population including mutational and splice variant ARs. Prostate Cancer Phase 2 Clinical
References References 1. Antonarakis ES, et al. Oncologist. 2016 Dec;21(12):1427-1435. View Related Products by Target Estrogen Receptor/ERR Prostate Cancer

 Chemical & Physical Properties

Molecular Formula C23H29ClO6
Molecular Weight 436.929