Epertinib hydrochloride
Modify Date: 2024-01-08 14:03:22
Epertinib hydrochloride structure
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Common Name | Epertinib hydrochloride | ||
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| CAS Number | 2071195-74-7 | Molecular Weight | 596.48 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C30H28Cl2FN5O3 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of Epertinib hydrochlorideEpertinib hydrochloride is a potent, orally active, reversible, and selective tyrosine kinase inhibitor of EGFR, HER2 and HER4, with IC50s of 1.48 nM, 7.15 nM and 2.49 nM, respectively. Epertinib shows potent antitumor activity[1]. |
| Name | Epertinib hydrochloride |
|---|
| Description | Epertinib hydrochloride is a potent, orally active, reversible, and selective tyrosine kinase inhibitor of EGFR, HER2 and HER4, with IC50s of 1.48 nM, 7.15 nM and 2.49 nM, respectively. Epertinib shows potent antitumor activity[1]. |
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| Related Catalog | |
| Target |
EGFR:1.48 nM (IC50) HER4:2.49 nM (IC50) HER2:7.15 nM (IC50) |
| References |
| Molecular Formula | C30H28Cl2FN5O3 |
|---|---|
| Molecular Weight | 596.48 |