BMS-212 structure
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Common Name | BMS-212 | ||
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CAS Number | 2173153-38-1 | Molecular Weight | 611.621 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C25H30N3O9PS2 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of BMS-212BMS-212 is a potent and selective stimulator of glucokinase (GK) (EC50 = 35 nM) that is promisingly used as an antidiabetic. |
Name | BMS-212 |
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Description | BMS-212 is a potent and selective stimulator of glucokinase (GK) (EC50 = 35 nM) that is promisingly used as an antidiabetic. |
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In Vitro | BMS-212 is a potent and selective stimulator of glucokinase (GK) (EC50 = 35 nM) that is promisingly used as an antidiabetic. BMS-212 has a preference for GK in liver over GK in pancreas, of which the activation may lead to non-glucose-dependent insulin secretion. Half-life of BMS-212 is 4.2h, and oral bioavailability is 15%. |
Molecular Formula | C25H30N3O9PS2 |
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Molecular Weight | 611.621 |