FR252384

Modify Date: 2024-01-10 17:42:25

FR252384 Structure
FR252384 structure
Common Name FR252384
CAS Number 447405-11-0 Molecular Weight 275.35
Density N/A Boiling Point N/A
Molecular Formula C18H17N3 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of FR252384


FR252384 is a neuropeptide Y-Y5 receptor antagonist, with an IC50 of 2.3 nM.

 Names

Name FR252384

 FR252384 Biological Activity

Description FR252384 is a neuropeptide Y-Y5 receptor antagonist, with an IC50 of 2.3 nM.
Related Catalog
Target

IC50: 2.3 nM (neuropeptide Y-Y5 receptor)[1]

In Vivo FR252384 is orally absorbable and permeable to brain[1].
References

[1]. Satoh Y, et al. Novel potent antagonists of human neuropeptide Y-Y5 receptor. Part 4: tetrahydrodiazabenzazulene derivatives. Bioorg Med Chem Lett. 2002 Apr 8;12(7):1009-11.

 Chemical & Physical Properties

Molecular Formula C18H17N3
Molecular Weight 275.35